• A prodrug is a pharmacologically inactive medication or compound that, after intake, is metabolized (i.e., converted within the body) into a pharmacologically...
    12 KB (1,279 words) - 13:32, 23 February 2024
  • Directed enzyme prodrug therapy (DEPT) uses enzymes artificially introduced into the body to convert prodrugs, which have no or poor biologically activity...
    12 KB (1,494 words) - 15:48, 29 August 2023
  • Thumbnail for Norethisterone
    estrogen in such research. However, NETE, an intramuscularly administered prodrug of norethisterone which is used as a long-acting contraceptive, is used...
    91 KB (9,305 words) - 06:23, 9 February 2024
  • Thumbnail for GABA analogue
    (γ-hydroxybutyric acid acetate) – synthetic prodrug to GHB GBL (γ-hydroxybutyric acid lactone) – metabolic intermediate and prodrug to GHB GHBAL (γ-hydroxybutyraldehyde...
    8 KB (754 words) - 04:40, 27 January 2024
  • called prodrugs. The reasons for this type of formulation may be because the drug is more stable during manufacture and storage as the prodrug form, or...
    4 KB (470 words) - 20:52, 9 January 2023
  • Thumbnail for Mometasone
    of mometasone, is the marketed medication. Mometasone furoate acts as a prodrug of mometasone. In addition to its glucocorticoid activity, mometasone also...
    31 KB (2,581 words) - 01:51, 31 March 2024
  • Hypoxia-Activated Prodrugs (HAPs) are prodrugs that target regions of tumor hypoxia within tumor cells. HAPs may offer the potential, alone and in combination...
    3 KB (372 words) - 10:09, 28 February 2022
  • Thumbnail for O-Acetylpsilocin
    O-Acetylpsilocin (category Prodrugs)
    psilocybin for pharmacological studies, as they are both believed to be prodrugs of psilocin. However, some users report that O-acetylpsilocin's subjective...
    12 KB (1,169 words) - 10:09, 24 February 2024
  • Thumbnail for Corticosteroid
    Corticosteroids are a class of steroid hormones that are produced in the adrenal cortex of vertebrates, as well as the synthetic analogues of these hormones...
    41 KB (4,133 words) - 04:03, 1 May 2024
  • Thumbnail for Boldenone undecylenate
    damage. Boldenone undecylenate is an androgen ester and a long-lasting prodrug of boldenone in the body. Boldenone undecylenate was introduced for medical...
    12 KB (870 words) - 22:35, 30 December 2023