 | pharmacology, GABAA receptor positive allosteric modulators, also known as GABAkines or GABAA receptor potentiators, are positive allosteric modulator (PAM) molecules... 31 KB (3,523 words) - 16:44, 26 April 2024 |
D1 receptor positive modulators. Allosteric regulation AMPA receptor positive allosteric modulator GABAA receptor positive allosteric modulator GABAA receptor... 19 KB (2,273 words) - 12:18, 26 August 2023 |
 | AMPA receptor positive allosteric modulators are positive allosteric modulators (PAMs) of the AMPA receptor (AMPR), a type of ionotropic glutamate receptor... 12 KB (1,256 words) - 01:39, 20 November 2023 |
A GABAA receptor negative allosteric modulator is a negative allosteric modulator (NAM), or inhibitor, of the GABAA receptor, a ligand-gated ion channel... 10 KB (934 words) - 07:32, 16 September 2023 |
 | Benzodiazepines like diazepam and midazolam act as positive allosteric modulators for GABAA receptors. When these receptors are activated, there's a rise in intracellular... 54 KB (5,992 words) - 15:58, 28 March 2024 |
A receptor modulator, or receptor ligand, is a general term for a substance, endogenous or exogenous, that binds to and regulates the activity of chemical... 8 KB (982 words) - 17:21, 11 April 2024 |
 | Zuranolone (category GABAA receptor positive allosteric modulators) inhibitory pregnane neurosteroid, zuranolone acts as a positive allosteric modulator of the GABAA receptor. Zuranolone was approved for medical use in the United... 16 KB (1,167 words) - 17:36, 5 March 2024 |
 | Alpidem (category GABAA receptor positive allosteric modulators) Z-drug zolpidem, and acts as a GABAA receptor positive allosteric modulator of the benzodiazepine site of the receptor complex. In contrast to zolpidem... 49 KB (4,669 words) - 06:29, 5 January 2024 |
 | Etifoxine (category GABAA receptor positive allosteric modulators) sedation or lack of coordination. Etifoxine acts as a GABAA receptor positive allosteric modulator and as a ligand for translocator proteins. Both mechanisms... 38 KB (3,481 words) - 20:48, 28 February 2024 |
 | Etizolam (category GABAA receptor positive allosteric modulators) its mode of action via the benzodiazepine receptor and directly targeting GABAA allosteric modulator receptors. It possesses anxiolytic, amnesic, anticonvulsant... 31 KB (2,765 words) - 18:59, 21 March 2024 |