= 98% E-6837 – Full agonist at human 5HT6 receptors E-6801 E-6837 – partial agonist at rat 5-HT6 receptors. Orally active in rats, and caused weight loss...
29 KB (3,301 words) - 21:37, 9 March 2024
which activates 5-HT1A, 5-HT1D, 5-HT1B, D2 and norepinephrine receptors. LSD (a psychedelic) is a 5-HT1A, 5-HT2A, 5-HT2C, 5-HT5A and 5-HT6 agonist. The genes...
65 KB (5,263 words) - 05:49, 28 March 2024
5-HT2A receptor 5-HT2B receptor 5-HT2C receptor 5-HT1 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Category:5-HT2...
2 KB (166 words) - 00:47, 13 May 2022
a 5-HT5A receptor agonist, and this action could be involved in the sleep-promoting effects of valerian. No selective agonists of the 5-HT6 receptor have...
16 KB (1,657 words) - 17:23, 8 June 2024
of 5-HT3 receptors in cell lines and native tissues quickly followed. 5-HT1 receptor 5-HT2 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7...
22 KB (2,391 words) - 07:50, 12 March 2024
nM) 5-HT2A receptors (Ki = 295 nM) 5-HT2B receptors (Ki = 16.4 nM) 5-HT2C receptors (Ki = 52.48 nM) 5-HT4 receptors (Ki = 501.18 nM) 5-HT6 receptors (Ki...
7 KB (619 words) - 21:37, 9 March 2024
Chamomile (ethanol extract) 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
18 KB (2,074 words) - 04:08, 7 May 2024
articles of the individual subtypes: 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Hoyer D, Clarke DE, Fozard JR...
5 KB (472 words) - 12:54, 25 December 2023
Paliperidone Risperidone 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor GRCh38: Ensembl release...
25 KB (2,990 words) - 04:12, 19 February 2024
The 5-HT2A receptor is a subtype of the 5-HT2 receptor that belongs to the serotonin receptor family and is a G protein-coupled receptor (GPCR). The 5-HT2A...
88 KB (9,594 words) - 07:13, 3 June 2024